产品编号：4083769

纯度规格：The MK2a Inhibitor, also referenced under CAS 41179-33-3, controls the biological activity of MK2a. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.

包装规格：5 MG

产品编号：4083768

纯度规格：The JNK Inhibitor VIII, also referenced under CAS 894804-07-0, controls the biological activity of JNK. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.

包装规格：5 MG

产品编号：4083767

纯度规格：The IP6K Inhibitor, also referenced under CAS 519178-28-0, controls the biological activity of IP6K.

包装规格：5 MG

产品编号：4083765

纯度规格：The Cdk9 Inhibitor II, also referenced under CAS 140651-18-9, controls the biological activity of Cdk9. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.

包装规格：5 MG

产品编号：4083764

纯度规格：The Cdk4 Inhibitor III, also referenced under CAS 265312-55-8, controls the biological activity of Cdk4. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.

包装规格：5 MG

产品编号：4083763

纯度规格：The Cdk4 Inhibitor II, NSC 625987, also referenced under CAS 141992-47-4, controls the biological activity of Cdk4. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.

包装规格：5 MG

产品编号：4083762

纯度规格：The Cdk2/9 Inhibitor, also referenced under CAS 507487-89-0, controls the biological activity of Cdk2/9. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.

包装规格：5 MG

产品编号：4083761

纯度规格：The Cathepsin L Inhibitor II controls the biological activity of Cathepsin L. This small molecule/inhibitor is primarily used for Protease Inhibitors applications.

包装规格：5 MG

产品编号：4083760

纯度规格：The Casein Kinase II Inhibitor III, TBCA, also referenced under CAS 934358-00-6, controls the biological activity of Casein Kinase II. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.

包装规格：5 MG

产品编号：4083759

纯度规格：A boronic acid-based arginine analog that acts as a slow-binding, competitive transition state inhibitor of arginases I and II (K_i = 310 nM for human recombinant type II arginase, pH 7.5).

包装规格：5 MG

产品编号：4083752

纯度规格：A cell-permeable, highly potent antagonist of TRPM8 (IC₅₀ = 10.9 nM in icilin evoked Ca2+ currents in HEK293 cells)

包装规格：10 MG

产品编号：4083751

纯度规格：A cell-permeable, active-site directed, acyl-donor substrate competitive inhibitor of transglutaminase 2 (TG2, K_i = 11 μM).

包装规格：5 MG

产品编号：4083750

纯度规格：Inhibits TNFα/β-stimulated biological activity by modulating, but not abolishing, TNF-TNFR interaction via direct TNF affinity interaction (KD = 110 nM).

包装规格：10 MG

产品编号：4083748

纯度规格：A cell-permeable, selective, highly potent, non-nucleotide competitive inhibitor of telomerase activity (IC₅₀ = 93 nM in HeLa cells nuclear extracts).

包装规格：10 MG

产品编号：4083747

包装规格：5 MG

产品编号：4083745

包装规格：10 MG

产品编号：4083744

包装规格：500 μG

产品编号：4083743

纯度规格：A cell-permeable, brain permeant, potent, reversible, ATP competitive inhibitor of Cdk4 and Cdk6 (IC₅₀ = 11, 9, and 15 nM for Cdk4/D1, Cdk4/D3 and Cdk6/D2, respectively).

包装规格：5 MG

产品编号：4083741

纯度规格：A cell permeable, selective, sphingosine competitive inhibitor of spingosine Kinase -2 (IC₅₀ = 4.3 μM).

包装规格：10 MG

产品编号：4083740

纯度规格：A peptidyl toxin from venom of African tarantula, Hysterocrates gigas that acts as a high affinity, reversible blocker of Cav2.3 (α1E, R-type) channels (IC₅₀ = 15-30 nM).

包装规格：10 μG

产品编号：4083738

纯度规格：A cell-permeable inhibitor of SKP2-dependent p27Kip1 ubiquitination. Selectively induces the accumulation SCFSKP2 substrates in multiple myeloma RPMI 8226 cells.

包装规格：10 MG

产品编号：4083737

包装规格：10 MG

产品编号：4083736

纯度规格：A highly potent agonist of GABAB receptor. Shown to be about 10-times more potent than baclofen.

包装规格：10 MG

产品编号：4083734

包装规格：10 MG

产品编号：4083725

纯度规格：A cell-permeable racemic mixture of Halofuginone that inhibits of prolyl-tRNA synthetase.

包装规格：10 MG

产品编号：4083724

纯度规格：A cell-permeable, selective inhibitor of protein arginine methyltransferase 1 (PRMT1; IC₅₀ = 9.5 μM).

包装规格：10 MG

产品编号：4083722

包装规格：10 MG

产品编号：4083721

纯度规格：A cell-permeable inhibitor of Wnt secretion from L-cell Wnt1/2/3/3a/6/7a/9a transfectants (IC₅₀ from 50 pM to 1.1 nM).

包装规格：5 MG

产品编号：4083717

纯度规格：A rhodanine-derived, reversible, photoactivated, TrpA1-selective channel activator.

包装规格：10 MG

产品编号：4083714

纯度规格：A cell-permeable, highly potent and selective inhibitor of phosphodiesterase 5 (PDEV; IC₅₀ = 270 pM).

包装规格：5 MG

产品编号：4083710

纯度规格：A cell-permeable compound that selectively downregulates the expression of p21 (~10 μM), independent of p53.expression, at either transcription or post-transcriptional level.

包装规格：10 MG

产品编号：4083706

纯度规格：A cell-permeable myristoylated hexapeptide that selectively inhibits integrin outside-in signaling without affecting inside-out signaling. Blocks the interaction of Gα3 and integrin β3 subunit.

包装规格：10 MG

产品编号：4083701

纯度规格：A cell-permeable. Reversible, selective inhibitor of the growth of malignant peripheral nerve sheath tumors (EC₅₀ = 439 nM, 754 nM, and 1.0 μM in S462, SNF96.2, and sMPNST cells).

包装规格：25 MG

产品编号：4083697

包装规格：10 MG

产品编号：4083692

纯度规格：A cell-permeable, potent, selective, reversible inhibitor of Lysine-Specific Demethylase 1 (LSD1; IC₅₀ = 13 nM; K_i = 31 nM).

包装规格：10 MG

产品编号：4083691

纯度规格：A cell-permeable, both NADH and pyruvate-competitive isoform A-selective LDH inhibitor. Exhibits enhanced anticancer activity under hypoxic conditions.

包装规格：10 MG

产品编号：4083690

纯度规格：A cell-permeable, fast acting, branched polyamine. Induces growth of actin-enriched lamellipodia within minutes without the need for serum cofactors .

包装规格：10 MG

产品编号：4083688

纯度规格：A voltage gated calcium channel gating inhibitor of the dihydropyridine class.

包装规格：10 MG

产品编号：4083686

纯度规格：A substrate competitive inhibitor of insulin-regulated aminopeptidase (IRAP) activity (K_i = 0.48 μM against 25 μM Leu-AMC).

包装规格：10 MG

产品编号：4083685

纯度规格：A 10 mM (5 mg/1.07 ml) sterile-filtered solution of Wnt Antagonist II, IWP-2) in DMSO.

包装规格：5 MG

产品编号：4083683

纯度规格：A 25 mM (5 mg/357 μl) sterile-filtered solution of PPACK, 2HCl in H₂O.

包装规格：5 MG

产品编号：4083680

包装规格：10 MG

产品编号：4083678

纯度规格：A 50 mM sterile-filtered solution of I-BET in DMSO.

包装规格：5 MG

产品编号：4083677

纯度规格：A 25 mM (2 mg/231 μl) sterile-filtered solution of Ginkgolic Acid (15:1) in DMSO.

包装规格：2 MG

产品编号：4083676

包装规格：5 MG

产品编号：4083675

包装规格：2 MG

产品编号：4083674

纯度规格：A 25 mM solution of (+)-Brefeldin A in DMSO.

包装规格：2 MG

产品编号：4083672

纯度规格：A cell-permeable compound that competitively binds to Hu antigen R (HuR; K_i = 350 nM) and disrupts the interaction of HuR and adenine- and uridine-rich element (ARE) of target mRNAs.

包装规格：10 MG

产品编号：4083670

包装规格：10 MG

产品编号：4083667

纯度规格：Cell-permeable inhibitor of gp130. Binds to gp130 and induces its phosphorylation at Ser782 in ovarian cancer cells. Suppresses constitutive phosphorylation of and nuclear translocation of Stat3.

包装规格：10 MG