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PKG Inhibitor-Calbiochem
| 产品编号： | 4061735 |
| 规格： | The PKG Inhibitor controls the biological activity of PKG. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications. |
| 包装规格： | 1 MG |
| 产品类别： | 进口试剂 |
| 品牌： | Sigma-Aldrich |
| 优惠价： | 立即咨询 |
产品别名
PKG Inhibitor-Calbiochem
Protein Kinase G Inhibitor, RKRARKE
基本信息
| Empirical Formula【经验(实验)分子式】 | C38H74N18O10 |
| Molecular weight | 943.11 |
| General description【一般描述】 | A specific, reversible, and substrate competitive inhibitor of PKG (Ki = 86 µM) relative to PKA (Ki = 550 µM). Sequence corresponds to a non-phosphorylatable analog (Ser32 to Ala32) of histone H2B (amino acids 29-35). A more specific, reversible, and substrate competitive inhibitor of protein kinase G (Ki = 86 µM) relative to protein kinase A (Ki = 550 µM). Sequence corresponds to a non-phosphorylatable analog (Ser32 to Ala32) of histone H2B (amino acids 29-35). |
| Biochem/physiol Actions【生化/生理作用】 | Target Ki: 86 µM against protein kinase G Product does not compete with ATP. Cell permeable: no Reversible: yes |
| Warning【警告】 | Toxicity: Standard Handling (A) |
| Sequence【序列】 | H-Arg-Lys-Arg-Ala-Arg-Lys-Glu-OH |
| Other Notes【其他说明】 | Glass, D.B., et al. 1983. Biochem. J.213, 159. |
| Legal Information【法律信息】 | CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany |
产品性质
| Quality Level【质量水平】 | 100 |
| Assay【测定】 | ≥95% (HPLC) |
| form【形式】 | lyophilized |
| manufacturer/tradename | Calbiochem® |
| storage condition【储存条件】 | OK to freeze desiccated (hygroscopic) |
| solubility【溶解性】 | water: 1 mg/mL |
| shipped in【运输】 | ambient |
| storage temp.【储存温度】 | −20℃ |
| packaging【包装】 | 1 mg in Plastic ampoule Yes |
安全信息
| Storage Class Code【储存分类代码】 | 11 - Combustible Solids |
| WGK | WGK 3 |
